Cytochrome P450 3a4 And 3a5 Known Drug Interaction Chart
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2Cytochrome P450 3A4 and 3A5 Known Drug Interaction Chart
CYP3A4 and CYP3A5 Inhibitors
CYP3A4 and CYP3A5 Substrates
ANTIHISTAMINES
NEUROPSYCHIATRIC
STRONG INHIBITORS
astemizole
alprazolam
clarithromycin
chlorpheniramine
diazepam
indinavir
ANTIMETRIC
midazolam
itraconazole
aprepitant
triazolam
ketoconazole
ondansetron
haloperidol
nefazodone
ANESTHESIA/PAIN
aripiprazole
ritonavir
cafergot
buspirone
saquinavir
codeine-N-demethylation
carbamazepine
suboxone
fentanyl
pimozide
telithromycin
levolevomethadyl acetate (LAAM)
quetiapine
INTERMEDIATE STRENGTH INHIBITORS
lidocaine,
risperidone
aprepitant
methadone
trazodone
erythromycin
ANTIBIOTIC/ANTIVIRAL
zaleplon
fluconazole
alfentanil
ziprasidone
grapefruit juice
boceprevir
zolpidem
verapamil
clarithromycin
ONCOLOGY
diltiazem
efavirenz
docetaxel
WEAK INHIBITORS
erythromycin (not CYP3A5),
gleevec
cimetidine
indinavir
irinotecan
OTHER POSSIBLE INHIBITORS
paclitaxel
nelfinavir
amiodarone
nevirapine
romidepsin
boceprevir
quinine
sorafenib
chloramphenicol
ritonavir
sunitinib
ciprofloxacin
saquinavir
torisel
delaviridine
telaprevir
vemurafenib
diethyl-dithiocarbamate
telithromycin.
vincristine
fluvoxamine
CARDIOVASCULAR
PULMONARY
gestodene
amlodipine
salmeterol
imatinib
cilostazol
sildenafil
mibefradil
diltiazem
STEROID
mifepristone
eplerenone
dexamethasone
norfloxacin
lercanidipine
estradiol
norfluoxetine
nifedipine
hydrocortisone
starfruit
nisoldipine
progesterone
telaprevir
nitrendipine
testosterone
voriconazole
propranolol
OTHER
quinidine (not CYP3A5)
cocaine
verapamil
dapsone
HMG COA REDUCTASE INHIBITORS
dextromethorphan
atorvastatin
finasteride
lovastatin
nateglinide
simvastatin
IMMUNE MODULATORS
cyclosporine
sirolimus
tacrolimus
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